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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
AS1517499 Influence on protin activity Western Blot 10.00 nM 264.7 RAW Mus musculus p-STAT6
AS1517499 Influence on protin activity Western Blot 100.00 nM 264.7 RAW Mus musculus p-STAT6
AS1517499 Influence on protin activity Western Blot 250.00 nM 264.7 RAW Mus musculus p-STAT6
AS1517499 Influence on protin activity Western Blot 10.00 nM 264.7 RAW Mus musculus STAT6
AS1517499 Influence on protin activity Western Blot 100.00 nM 264.7 RAW Mus musculus STAT6
AS1517499 Influence on protin activity Western Blot 250.00 nM 264.7 RAW Mus musculus STAT6
AS1517499 Influence on protin activity Western Blot 10.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on protin activity Western Blot 100.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on protin activity Western Blot 250.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 10.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 100.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 250.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 10.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 100.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 250.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 10.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 100.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 250.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 10.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 100.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on macrophage differentiation RT-qPCR 250.00 nM 264.7 RAW Mus musculus
AS1517499 Influence on cell viability Resazurin sodium salt 100.00 nM 4T1-luc Mus musculus
AS1517499 Influence on cell viability Resazurin sodium salt 250.00 nM 4T1-luc Mus musculus
AS1517499 Influence on cell proliferation in tumor tissue Tumor volume 20.00 mg/kg 4T1-luc (xenograft) Mus musculus BALB/c
AS1517499 Influence on cell proliferation in tumor tissue IVIS in vivo imaging 20.00 mg/kg 4T1-luc (xenograft) Mus musculus BALB/c
AS1517499 Influence on tumor metastasis IVIS in vivo imaging 20.00 mg/kg liver Mus musculus BALB/c
AS1517499 Influence on tumor progression RT-qPCR 20.00 mg/kg macrophages Mus musculus BALB/c
AS1517499 Influence on tumor progression RT-qPCR 20.00 mg/kg macrophages Mus musculus BALB/c
AS1517499 Influence on tumor progression RT-qPCR 20.00 mg/kg macrophages Mus musculus BALB/c
AS1517499 Influence on tumor progression RT-qPCR 20.00 mg/kg liver Mus musculus BALB/c
AS1517499 Influence on tumor progression RT-qPCR 20.00 mg/kg liver Mus musculus BALB/c
AS1517499 Influence on tumor progression RT-qPCR 20.00 mg/kg liver Mus musculus BALB/c
AS1517499 Influence on protein activity 2 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6 p-STAT6 (Y641)
AS1517499 Influence on protein activity 2 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6 STAT6
AS1517499 Influence on protein activity 2 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6
AS1517499 Influence on protein activity 7 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6 p-STAT6 (Y641)
AS1517499 Influence on protein activity 7 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6 STAT6
AS1517499 Influence on protein activity 7 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6
AS1517499 Influence on protein activity 14 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6 p-STAT6 (Y641)
AS1517499 Influence on protein activity 14 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6 STAT6
AS1517499 Influence on protein activity 14 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6
AS1517499 Influence on protein activity 2 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6
AS1517499 Influence on protein activity 2 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6
AS1517499 Influence on protein activity 7 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6
AS1517499 Influence on protein activity 14 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6
AS1517499 Influence on protein activity 14 days post-bleomycin treatment Western Blot 10.00 mg/kg lung tissue Mus musculus c57BL/6
AS1517499 Influence on protein activity 7 days post-bleomycin treatment Immuinofluorescence 10.00 mg/kg alveolar macrophages Mus musculus c57BL/6
AS1517499 Influence on protein activity 2 days post-bleomycin treatment Immuinofluorescence 10.00 mg/kg alveolar macrophages Mus musculus c57BL/6
AS1517499 Influence on STAT6 dependent genes RT-qPCR 10.00 mg/kg alveolar macrophages Mus musculus c57BL/6
AS1517499 Influence on STAT6 dependent genes RT-qPCR 10.00 mg/kg lung tissue Mus musculus c57BL/6